To determine the given K I and I50 values. Whether the compound A is effective in preventing HIV replication when taken orally or not should be determined. Concept introduction: The IC50, half maximal inhibitory concentration, is the capacity of a substance to inhibit biological molecules and biochemical reactions. IC50 is the quantitative measurement of the inhibitor, which indicates the amount of inhibitor required to inhibit the biological substance.

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Chapter 28, Problem 14P

Interpretation Introduction

Interpretation:

To determine the given K_I and I50 values. Whether the compound A is effective in preventing HIV replication when taken orally or not should be determined.

Concept introduction:

The IC50, half maximal inhibitory concentration, is the capacity of a substance to inhibit biological molecules and biochemical reactions. IC50 is the quantitative measurement of the inhibitor, which indicates the amount of inhibitor required to inhibit the biological substance.

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