Choose (+) if the following circumstances or situations will most likely result to production of intrinsic activity; if otherwise, choose (-) Choose (+) if the following circumstances or situations will most likely result to production of intrinsicactivity; if otherwise, choose (-).+Dissociation of drugmolecule from binding siteFormation of H-bondsbetween drug and receptorPresence of hydrophobicinteractionsIntroduction of an antagonistat receptor sitesHigh concentration ofcompetitive antagonist at thebinding siteBlockade of binding site dueto steric hindranceComplementing shapes ofdrug and binding siteLack of affinity between drugand binding siteFormation of an irreversibledrug-receptor complexConformational changebetween drug and receptorafter binding

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Choose (+) if the following circumstances or situations will most likely result to production of intrinsic activity, if otherwise, choose (-). Dissociation of drug molecule from binding site

Biochemistry

9th Edition

ISBN:9781319114671

Author:Lubert Stryer, Jeremy M. Berg, John L. Tymoczko, Gregory J. Gatto Jr.

Publisher:Lubert Stryer, Jeremy M. Berg, John L. Tymoczko, Gregory J. Gatto Jr.

Chapter1: Biochemistry: An Evolving Science

Section: Chapter Questions

Problem 1P

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