All of the following are reasons for considering the enzymes as druggable targets except: enzymes have the allosteric sites where modulators can bind it is easy to purify in significant amount and characterize the enzymes enzyme kinetics concepts are well established for identifying inhibitors and activators hits and leads can be identified from known substrates and transition-states

All of the following are reasons for considering the enzymes as druggable targets except: enzymes have the allosteric sites where modulators can bind it is easy to purify in significant amount and characterize the enzymes enzyme kinetics concepts are well established for identifying inhibitors and activators hits and leads can be identified from known substrates and transition-states

Chemistry

10th Edition

ISBN:9781305957404

Author:Steven S. Zumdahl, Susan A. Zumdahl, Donald J. DeCoste

Publisher:Steven S. Zumdahl, Susan A. Zumdahl, Donald J. DeCoste

Chapter1: Chemical Foundations

Section: Chapter Questions

Problem 1RQ: Define and explain the differences between the following terms. a. law and theory b. theory and...

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